平安! 发表于 2011-11-9 19:57
) y j W( V. o# J% y* vPazopanib (100 mg/kg/day free base equivalent)
# h) \5 l" u1 ~! h. g3 d9 m% \ 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。& J: a% Y9 _% C/ J W8 X
搜索了一下,原料一大堆。: D+ G/ Q" j1 }5 {4 z9 g! w
& B1 S L% H P+ K- b8 h2 M' l4 D! i! C对不起!100mg/kg是用于移植瘤的,我弄错了。
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以下是正版说明书的推荐用量。/ I" U/ N& Q% L% O$ z
+ K6 d" _ a- c8 o+ C--------------------- DOSAGE AND ADMINISTRATION ----------------+ N, U4 F$ X4 @4 o
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) k: i7 c" H; W
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) 9 c0 b6 O$ V, _7 M/ S6 p
---------------------DOSAGE FORMS AND STRENGTHS --------------) I* I2 u. e. N' J% O( B
200 mg tablets. (3)
: t. ~' [9 J; n/ O-------------------------------CONTRAINDICATIONS------------------------ |