平安! 发表于 2011-11-9 19:57 ! @/ J! ?! o/ j+ B- S
Pazopanib (100 mg/kg/day free base equivalent)
g0 V5 a* T. }5 O9 ]9 e# R 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。& |: M% z% ]% B: i* L) H# M* i6 y
搜索了一下,原料一大堆。( {+ ^9 U* @3 k5 v7 O5 h i/ ]
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对不起!100mg/kg是用于移植瘤的,我弄错了。: q. ?' _# d8 c3 u) R8 E1 G
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以下是正版说明书的推荐用量。
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--------------------- DOSAGE AND ADMINISTRATION ----------------
! @- u% M% d# i* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
( c3 N* C8 S4 W, w+ r" W* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
8 T: y7 o3 s3 j$ k6 Q0 u---------------------DOSAGE FORMS AND STRENGTHS --------------" @! ^2 U$ a+ u( B
200 mg tablets. (3) ( J, t P: M3 Y9 A
-------------------------------CONTRAINDICATIONS------------------------ |