平安! 发表于 2011-11-9 19:57 6 m9 z2 G$ E; x1 y/ N
Pazopanib (100 mg/kg/day free base equivalent)
; x3 b# i- Y% | 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。; h) O- t4 I, u# G
搜索了一下,原料一大堆。
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对不起!100mg/kg是用于移植瘤的,我弄错了。6 |- }1 A1 g+ W# R
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以下是正版说明书的推荐用量。0 q7 y( c6 Z( ~: p
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--------------------- DOSAGE AND ADMINISTRATION ----------------
4 \* Z/ S& S. l; R5 Z* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) % s2 v" E" L. n* X9 C" K; J
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) 1 s9 a' b, `- w s S
---------------------DOSAGE FORMS AND STRENGTHS --------------& F# Q$ i5 A! Y5 F6 `0 d
200 mg tablets. (3) M C7 e4 p, ?% ^- ^' H) y* Z4 s
-------------------------------CONTRAINDICATIONS------------------------ |